BDBM50233224 CHEMBL4070670
SMILES CCCCCCCCCC[C@H]1C[C@@]2(CCCO2)NC(=N)N1
InChI Key InChIKey=NODTXKHXBIVQCH-RDJZCZTQSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50233224
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human Nav1.2 expressed in HEK293T cells assessed as inhibition of VTD-induced tail current by whole cell patch clamp method re...More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human Nav1.2 expressed in HEK293T cells assessed as inhibition of VTD-induced sustained current by whole cell patch clamp meth...More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Inhibition of Nav1.2 (unknown origin) by cell based assayMore data for this Ligand-Target Pair