BDBM50235763 (2R,3R)-methyl 2-(1-(2-((S)-1-amino-2-methylpropyl)-4-methylphenyl)piperazine-4-carbonyl)-3-(4-chlorophenyl)pyrrolidine-1-carboxylate::CHEMBL255100
SMILES COC(=O)N1CC[C@@H]([C@@H]1C(=O)N1CCN(CC1)c1ccc(C)cc1[C@@H](N)C(C)C)c1ccc(Cl)cc1
InChI Key InChIKey=QFNYNYUWRSANTP-ZSQFBXSQSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50235763
Affinity DataKi: 17nMAssay Description:Displacement of [125]NDPMSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [125]NDPMSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 720nMAssay Description:Antagonist activity at MC4 receptor assessed as inhibition of alpha-MSH-stimulated cAMP productionMore data for this Ligand-Target Pair