BDBM50243571 (2R)-2-amino-N-[(4R,7S,10S,13R,16S,19S)-10-(4-aminobutyl)-4-{[(1S)-1-carbamoyl-2-(naphthalen-2-yl)ethyl]carbamoyl}-7-[(1R)-1-hydroxyethyl]-13-(1H-indol-3-ylmethyl)-16-({4-[(methoxycarbamoyl)amino]phenyl}methyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaazacycloicosan-19-yl]-3-(4-chlorophenyl)propanamide::CHEMBL499760
SMILES CONC(=O)Nc1ccc(C[C@@H]2NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc3c[nH]c4ccccc34)NC2=O)[C@@H](C)O)C(=O)N[C@@H](Cc2ccc3ccccc3c2)C(N)=O)NC(=O)[C@H](N)Cc2ccc(Cl)cc2)cc1
InChI Key InChIKey=FAZJEADZIKXOCO-BPBSOZPZSA-N
Data 5 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50243571
Affinity DataIC50: 313nMAssay Description:Displacement of [125I][LTT]SRIF28 from human cloned sst5 receptor by autoradiographyMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][LTT]SRIF28 from human cloned sst1 receptor by autoradiographyMore data for this Ligand-Target Pair
Affinity DataIC50: 883nMAssay Description:Displacement of [125I][LTT]SRIF28 from human cloned sst4 receptor by autoradiographyMore data for this Ligand-Target Pair
Affinity DataIC50: 157nMAssay Description:Displacement of [125I][LTT]SRIF28 from human cloned sst3 receptor by autoradiographyMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30nMAssay Description:Displacement of [125I][LTT]SRIF28 from human cloned sst2 receptor by autoradiographyMore data for this Ligand-Target Pair