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BDBM50244993 4-(3-phenyl-1,2,4-thiadiazol-5-yl)-N-(pyridin-3-yl)piperazine-1-carboxamide::CHEMBL513553

SMILES: O=C(Nc1cccnc1)N1CCN(CC1)c1nc(ns1)-c1ccccc1

InChI Key: InChIKey=RCAFZHFLIBYWGO-UHFFFAOYSA-N

Data: 4 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50244993
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Fatty-acid amide hydrolase 1 (Human)	BDBM50244993 (4-(3-phenyl-1,2,4-thiadiazol-5-yl)-N-(pyridin-3-yl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	9.80	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Fatty-acid amide hydrolase 1 [30-579] (Rat)	BDBM50244993 (4-(3-phenyl-1,2,4-thiadiazol-5-yl)-N-(pyridin-3-yl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	8.70	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Fatty-acid amide hydrolase 1 [30-579] (Rat)	BDBM50244993 (4-(3-phenyl-1,2,4-thiadiazol-5-yl)-N-(pyridin-3-yl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.80	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Fatty-acid amide hydrolase 1 (Human)	BDBM50244993 (4-(3-phenyl-1,2,4-thiadiazol-5-yl)-N-(pyridin-3-yl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.40	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair