BDBM50247086 CHEMBL444970::Chlorphrifos oxon::diethyl 3,5,6-trichloropyridin-2-yl phosphate
SMILES CCOP(=O)(OCC)Oc1nc(Cl)c(Cl)cc1Cl
InChI Key InChIKey=OTMOUPHCTWPNSL-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 11 hits for monomerid = 50247086
TargetMuscarinic acetylcholine receptor DM1(Drosophila melanogaster)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]AF-DX 384 from Drosophila melanogaster mAChR by scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor DM1(Drosophila melanogaster)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]QNB from Drosophila melanogaster mAChR by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in mouse brainMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]CP55940 from mouse CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+4nMAssay Description:Displacement of [3H]CP55940 from mouse CB1 receptor expressed in HEK293 cells in presence of mouse brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of 2-arachidonylglycerol from MAGL in Swiss Webster mouse brain after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 460nMAssay Description:Displacement of [3H]anandamide from FAAH in Swiss Webster mouse brain after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Displacement of acetylcholine from AChE in Swiss Webster mouse brain after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of FAAH-mediated [3H]anadamide hydrolysis in mouse brainMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of MAGL-mediated 2-arachidonoylglycerol hydrolysis in mouse brainMore data for this Ligand-Target Pair
Affinity DataKd: 0.860nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in mouse brain at 100 nMMore data for this Ligand-Target Pair