BDBM50257761 (R)-methyl 1-((S)-2-(3-(3-aminopropanamido)phenylsulfonamido)-3-(3-carbamimidoylphenyl)propanoyl)piperidine-2-carboxylate::CHEMBL492333

SMILES COC(=O)[C@H]1CCCCN1C(=O)[C@H](Cc1cccc(c1)C(N)=N)NS(=O)(=O)c1cccc(NC(=O)CCN)c1

InChI Key InChIKey=DFJXDNJQGLNAPO-FCHUYYIVSA-N

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50257761   

TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257761((R)-methyl 1-((S)-2-(3-(3-aminopropanamido)phenyls...)
Affinity DataKi:  100nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257761((R)-methyl 1-((S)-2-(3-(3-aminopropanamido)phenyls...)
Affinity DataKi:  100nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257761((R)-methyl 1-((S)-2-(3-(3-aminopropanamido)phenyls...)
Affinity DataKi:  4.90E+3nMAssay Description:Inhibition of plasmin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257761((R)-methyl 1-((S)-2-(3-(3-aminopropanamido)phenyls...)
Affinity DataKi:  2.42E+4nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
The Medicines Company (Leipzig)

Curated by ChEMBL
LigandPNGBDBM50257761((R)-methyl 1-((S)-2-(3-(3-aminopropanamido)phenyls...)
Affinity DataKi:  7.60E+4nMAssay Description:Inhibition of uPA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed