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BDBM50263224 CHEMBL4066795

SMILES: C1C2=C(CN1)N(C(=O)NC2=O)C[C@@H](C(=O)O)N

InChI Key: InChIKey=PGFCMMRTCMWFGC-UHFFFAOYSA-N

Data: 4 KI

PDB links: 1 PDB ID matches this monomer.

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50263224
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Glutamate receptor ionotropic, kainate 1 (Rat)	BDBM50263224 (CHEMBL4066795) Show SMILES Show InChI	GoogleScholar	UniChem		869	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Glutamate receptor 2 (Rat)	BDBM50263224 (CHEMBL4066795) Show SMILES Show InChI	GoogleScholar	UniChem		2.37E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 3 (Rat)	BDBM50263224 (CHEMBL4066795) Show SMILES Show InChI	GoogleScholar	UniChem		1.81E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 2 (Rat)	BDBM50263224 (CHEMBL4066795) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+6	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair