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BDBM50267372 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide::1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-morpholino-1H-pyrazole-3-carboxamide::AM-281::CHEMBL476833
SMILES: Cc1c(nn(c1-c1ccc(I)cc1)-c1ccc(Cl)cc1Cl)C(=O)NN1CCOCC1
InChI Key: InChIKey=AJFFBPZYXRNAIC-UHFFFAOYSA-N
Data: 6 KI
| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Cannabinoid receptor 1 (Rat) | BDBM50267372![]() (AM-281 | 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4...) | GoogleScholar | UniChem | 12.4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cannabinoid receptor 1 (Human) | BDBM50267372![]() (AM-281 | 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4...) | GoogleScholar | UniChem | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cannabinoid receptor 1 (Human) | BDBM50267372![]() (AM-281 | 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4...) | GoogleScholar | UniChem | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cannabinoid receptor 1 (Human) | BDBM50267372![]() (AM-281 | 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4...) | GoogleScholar | UniChem | 422 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cannabinoid receptor 2 (Rat) | BDBM50267372![]() (AM-281 | 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4...) | GoogleScholar | UniChem | 4.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Cannabinoid receptor 2 (Human) | BDBM50267372![]() (AM-281 | 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4...) | GoogleScholar | UniChem | 4.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||