BDBM50274461 CHEMBL504587::FGGFTGARKSARKWANQ

SMILES C[C@@H](O)[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(O)=O

InChI Key InChIKey=MRPJNGQFWWZSQY-FMCSKRGOSA-N

Data  2 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50274461   

TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50274461(CHEMBL504587 | FGGFTGARKSARKWANQ)
Affinity DataIC50:  0.410nMAssay Description:Displacement of [3H]nociceptin from rat ORL1 receptor expressed in african green monkey COS7 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50274461(CHEMBL504587 | FGGFTGARKSARKWANQ)
Affinity DataEC50:  5.80nMAssay Description:Activation of rat ORL1 receptor expressed in african green monkey COS7 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50274461(CHEMBL504587 | FGGFTGARKSARKWANQ)
Affinity DataIC50:  0.410nMAssay Description:Displacement of [3H]nociceptin from rat ORL1 receptor expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(RAT)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50274461(CHEMBL504587 | FGGFTGARKSARKWANQ)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at rat ORL1 receptor expressed in african green monkey COS7 cells assessed as stimulation of [35S]GTPgammaS binding by radioligand r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed