BDBM50275819 CHEMBL4125837

SMILES COc1cc(cc(OC)c1NS(C)(=O)=O)C(C)C(=O)NCc1ccc(nc1N1CCC(C)CC1)C(F)(F)F

InChI Key InChIKey=MQCKIQPZGIHBFB-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50275819   

TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50275819(CHEMBL4125837)
Affinity DataKi:  1.60nMAssay Description:Antagonist activity at recombinant human TRPV1 expressed in CHOK1 cells assessed as reduction in capsaicin-induced Ca2+ flux after 15 mins by fluo-4-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed