BDBM50289879 CHEMBL62205::[(S)-2-(1H-Indol-3-yl)-1-methyl-1-phenethylcarbamoyl-ethyl]-carbamic acid adamantan-2-yl ester
SMILES C[C@@](Cc1c[nH]c2ccccc12)(NC(=O)OC1C2CC3CC(C2)CC1C3)C(=O)NCCc1ccccc1
InChI Key InChIKey=RGFJPHVCLXSEHE-GYSLRPEDSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50289879
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Affinity DataKi: 21.4nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in mouse cortex membraneMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 377nMAssay Description:In vitro inhibition of [125I]- Bolton Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreas.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:In vitro inhibition of [125I]- Bolton Hunter CCK-8 binding to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Compound was evaluated for the binding affinity towards rat pancreatic Cholecystokinin type A receptorMore data for this Ligand-Target Pair