BDBM50293262 2-(5-benzyl-2-hydroxyphenyl)-6-methylquinolin-4(1H)-one::CHEMBL502159

SMILES Cc1ccc2nc(cc(O)c2c1)-c1cc(Cc2ccccc2)ccc1O

InChI Key InChIKey=ZTLOBJCILUZKRV-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50293262   

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Lund University

Curated by ChEMBL
LigandPNGBDBM50293262(2-(5-benzyl-2-hydroxyphenyl)-6-methylquinolin-4(1H...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha1beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(RAT)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293262(2-(5-benzyl-2-hydroxyphenyl)-6-methylquinolin-4(1H...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha5beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Rattus norvegicus (Rat))
Lund University

Curated by ChEMBL
LigandPNGBDBM50293262(2-(5-benzyl-2-hydroxyphenyl)-6-methylquinolin-4(1H...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha2beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(RAT)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293262(2-(5-benzyl-2-hydroxyphenyl)-6-methylquinolin-4(1H...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha3beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed