BDBM50293263 2-(5-benzyl-2-hydroxyphenyl)-6-methyl-4H-chromen-4-one::CHEMBL522061

SMILES Cc1ccc2oc(cc(=O)c2c1)-c1cc(Cc2ccccc2)ccc1O

InChI Key InChIKey=UHHVZGAPCPFAGJ-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50293263   

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Lund University

Curated by ChEMBL
LigandPNGBDBM50293263(2-(5-benzyl-2-hydroxyphenyl)-6-methyl-4H-chromen-4...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha1beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(RAT)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293263(2-(5-benzyl-2-hydroxyphenyl)-6-methyl-4H-chromen-4...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha5beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(RAT)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293263(2-(5-benzyl-2-hydroxyphenyl)-6-methyl-4H-chromen-4...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha3beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Rattus norvegicus (Rat))
Lund University

Curated by ChEMBL
LigandPNGBDBM50293263(2-(5-benzyl-2-hydroxyphenyl)-6-methyl-4H-chromen-4...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha2beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed