BDBM50294063 (3aR,6aR)-4'-(5-Methyl-hexahydro-pyrrolo[3,4-b]pyrrol-1-yl)-biphenyl-4-carbonitrile::CHEMBL563998
SMILES CN1C[C@H]2CCN([C@H]2C1)c1ccc(cc1)-c1ccc(cc1)C#N
InChI Key InChIKey=CXRCFQKCULIFAC-QUCCMNQESA-N
Data 3 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50294063
Affinity DataKi: 0.540nMAssay Description:Displacement of [3H]N-alpha methyl histamine from human cloned histamine H3 receptor expressed in C6 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.57nMAssay Description:Displacement of [3H]N-alpha methyl histamine from rat cortical membrane histamine H3 receptorMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 282nMAssay Description:Binding affinity to human ERG channelMore data for this Ligand-Target Pair