BDBM50294253 (4R,7S,10S,13S,16S,19R)-19-amino-N-((2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl)-7,16-dibenzyl-10-(4-((isopropylamino)methyl)benzyl)-13-(N-methyl-2-naphthamido)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaazacycloicosane-4-carboxamide::CHEMBL563462
SMILES CC(C)NCc1ccc(C[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](Cc3ccccc3)NC(=O)[C@@H](N)CSSC[C@H](NC(=O)[C@H](Cc3ccccc3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(N)=O)N(C)C(=O)c2ccc3ccccc3c2)cc1
InChI Key InChIKey=VABWJEMMIDGNDC-SWDBKDPZSA-N
Data 5 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50294253
TargetSomatostatin receptor type 4(Homo sapiens (Human))
The Clayton Foundation Laboratories For Peptide Biology
Curated by ChEMBL
The Clayton Foundation Laboratories For Peptide Biology
Curated by ChEMBL
Affinity DataIC50: 525nMAssay Description:Displacement of [125I]LTT-SRIF-28 from human sst4 receptor by autoradiographyMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
The Clayton Foundation Laboratories For Peptide Biology
Curated by ChEMBL
The Clayton Foundation Laboratories For Peptide Biology
Curated by ChEMBL
Affinity DataIC50: 253nMAssay Description:Displacement of [125I]LTT-SRIF-28 from human sst3 receptor by autoradiographyMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
The Clayton Foundation Laboratories For Peptide Biology
Curated by ChEMBL
The Clayton Foundation Laboratories For Peptide Biology
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]LTT-SRIF-28 from human sst2 receptor by autoradiographyMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
The Clayton Foundation Laboratories For Peptide Biology
Curated by ChEMBL
The Clayton Foundation Laboratories For Peptide Biology
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Displacement of [125I]LTT-SRIF-28 from human sst1 receptor by autoradiographyMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
The Clayton Foundation Laboratories For Peptide Biology
Curated by ChEMBL
The Clayton Foundation Laboratories For Peptide Biology
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]LTT-SRIF-28 from human sst5 receptor by autoradiographyMore data for this Ligand-Target Pair