BDBM50303556 (1-((Tetrahydrofuran-3-yl)methyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone::CHEMBL569994

SMILES CC1(C)C(C(=O)c2cn(CC3CCOC3)c3ccccc23)C1(C)C

InChI Key InChIKey=RKJJVEGZZUFFPU-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50303556   

TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50303556((1-((Tetrahydrofuran-3-yl)methyl)-1H-indol-3-yl)(2...)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50303556((1-((Tetrahydrofuran-3-yl)methyl)-1H-indol-3-yl)(2...)
Affinity DataKi:  630nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50303556((1-((Tetrahydrofuran-3-yl)methyl)-1H-indol-3-yl)(2...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in HEK293 cells coexpressing Galphaq/o5 assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed