BDBM50303575 CHEMBL570907::Cyclopentyl(1-((tetrahydro-2H-pyran-4-yl)methyl)-1H-indol-3-yl)methanone

SMILES O=C(C1CCCC1)c1cn(CC2CCOCC2)c2ccccc12

InChI Key InChIKey=UKZQAPQRIDWZDG-UHFFFAOYSA-N

Data  4 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50303575   

TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50303575(CHEMBL570907 | Cyclopentyl(1-((tetrahydro-2H-pyran...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50303575(CHEMBL570907 | Cyclopentyl(1-((tetrahydro-2H-pyran...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP 55940 from human CB2 receptor in cell free systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50303575(CHEMBL570907 | Cyclopentyl(1-((tetrahydro-2H-pyran...)
Affinity DataKi:  131nMAssay Description:Displacement of [3H]CP 55940 from human CB1 receptor in cell free systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50303575(CHEMBL570907 | Cyclopentyl(1-((tetrahydro-2H-pyran...)
Affinity DataKi:  131nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50303575(CHEMBL570907 | Cyclopentyl(1-((tetrahydro-2H-pyran...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in HEK293 cells coexpressing Galphaq/o5 assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed