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BDBM50303587 1-(3-tert-butyl-1-m-tolyl-1H-pyrazol-5-yl)-3-(4-chlorophenyl)urea::CHEMBL568875

SMILES: Cc1cccc(c1)-n1nc(cc1NC(=O)Nc1ccc(Cl)cc1)C(C)(C)C

InChI Key: InChIKey=RYCUVZMYBSSMAE-UHFFFAOYSA-N

Data: 5 IC50 1 Kd

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50303587
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Mitogen-activated protein kinase 14 (Human)	BDBM50303587 (1-(3-tert-butyl-1-m-tolyl-1H-pyrazol-5-yl)-3-(4-ch...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Mitogen-activated protein kinase 9 (Human)	BDBM50303587 (1-(3-tert-butyl-1-m-tolyl-1H-pyrazol-5-yl)-3-(4-ch...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	440	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Mitogen-activated protein kinase 9 (Human)	BDBM50303587 (1-(3-tert-butyl-1-m-tolyl-1H-pyrazol-5-yl)-3-(4-ch...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Mitogen-activated protein kinase 14 (Human)	BDBM50303587 (1-(3-tert-butyl-1-m-tolyl-1H-pyrazol-5-yl)-3-(4-ch...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Discoidin domain-containing receptor 2 (Human)	BDBM50303587 (1-(3-tert-butyl-1-m-tolyl-1H-pyrazol-5-yl)-3-(4-ch...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	183	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Discoidin domain-containing receptor 2 (Human)	BDBM50303587 (1-(3-tert-butyl-1-m-tolyl-1H-pyrazol-5-yl)-3-(4-ch...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	15	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair