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BDBM50304820 2-(piperazin-1-yl)-5,6,7,8-tetrahydroquinoline::CHEMBL593547

SMILES: C1CCc2nc(ccc2C1)N1CCNCC1

InChI Key: InChIKey=OHJFBSROVXQKFQ-UHFFFAOYSA-N

Data: 2 KI 2 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50304820
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
5-hydroxytryptamine receptor 2C (Human)	BDBM50304820 (2-(piperazin-1-yl)-5,6,7,8-tetrahydroquinoline \| C...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	25	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 2A (Human)	BDBM50304820 (2-(piperazin-1-yl)-5,6,7,8-tetrahydroquinoline \| C...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	2.20E+3	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 2A (Rat)	BDBM50304820 (2-(piperazin-1-yl)-5,6,7,8-tetrahydroquinoline \| C...) Show SMILES Show InChI	GoogleScholar	UniChem		21	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 2C (Human)	BDBM50304820 (2-(piperazin-1-yl)-5,6,7,8-tetrahydroquinoline \| C...) Show SMILES Show InChI	GoogleScholar	UniChem		45	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair