BDBM50309072 CHEMBL592054::IMIGLITAZAR

SMILES Cc1oc(nc1COc1ccc(CO\N=C(/CCC(O)=O)c2ccccc2)cc1)-c1ccccc1

InChI Key InChIKey=ULVDFHLHKNJICZ-QCWLDUFUSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50309072   

TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309072(CHEMBL592054 | IMIGLITAZAR)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309072(CHEMBL592054 | IMIGLITAZAR)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human PPARgamma transactivation expressed in human HePG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309072(CHEMBL592054 | IMIGLITAZAR)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human PPARalpha transactivation expressed in human HePG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309072(CHEMBL592054 | IMIGLITAZAR)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed