BDBM50312425 2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid::CHEMBL1075682

SMILES Cc1cc(OCc2nc(c(s2)-c2ccc(OC(F)(F)F)cc2)-c2ccc(OC3CCCC3)cc2)ccc1OCC(O)=O

InChI Key InChIKey=BONJIRURBUJMTG-UHFFFAOYSA-N

Data  5 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50312425   

TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50312425(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human PPARdelta ligand binding domain by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50312425(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human PPARdelta ligand binding domain expressed in human 293T cells cotransfected with Gal4-DBD by luciferase transactivation ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50312425(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human 293T cells cotransfected with Gal4-DBD by luciferase transactivation ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50312425(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human 293T cells cotransfected with Gal4-DBD by luciferase transactivation ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50312425(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
Affinity DataEC50:  31nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed