BDBM50314000 3-(4-(2-fluorophenyl)piperazine-1-carbonyl)-8-mesityl-2-methyl-5,6-dihydroimidazo[1,2-a]pyrimidin-7(8H)-one::CHEMBL1088325

SMILES Cc1nc2N(C(=O)CCn2c1C(=O)N1CCN(CC1)c1ccccc1F)c1c(C)cc(C)cc1C

InChI Key InChIKey=ISYXQSJHBBCMFG-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50314000   

TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Research & Development

Curated by ChEMBL
LigandPNGBDBM50314000(3-(4-(2-fluorophenyl)piperazine-1-carbonyl)-8-mesi...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from human CRFR1 expressed in human IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed