BDBM50322143 3-(4-chlorophenylsulfonyl)-N-(2,3-dimethylphenyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine::CHEMBL1170687

SMILES Cc1cccc(Nc2nc3c(nnn3c3ccsc23)S(=O)(=O)c2ccc(Cl)cc2)c1C

InChI Key InChIKey=KWSRBKUWEMKUOG-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50322143   

Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50322143(3-(4-chlorophenylsulfonyl)-N-(2,3-dimethylphenyl)t...)
Affinity DataIC50:  800nMAssay Description:Antagonist activity at human recombinant 5HT6 receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed