BDBM50331016 6-benzyl-3-(pyridin-3-yl)-6-azabicyclo[3.2.2]non-2-ene::CHEMBL1277968
SMILES C(N1CC2CCC1CC(=C2)c1cccnc1)c1ccccc1
InChI Key InChIKey=CRKOAXCURNCJRQ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50331016
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataKi: 1.95nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK292 cells after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK292 cells after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataKi: 424nMAssay Description:Displacement of [3H]epibatidine from alpha7 nAChR in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataEC50: 2.00E+3nMAssay Description:Partial agonist activity at rat alpha3beta4 nAChR expressed in HEK292 cells assessed as increase of calcium influx by FLIPR assayMore data for this Ligand-Target Pair