BDBM50334491 3-(4-((3-cyclohexyl-1-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-4-yl)methyl)benzamido)propanoic acid::CHEMBL1644173

SMILES OC(=O)CCNC(=O)c1ccc(Cc2cn(nc2C2CCCCC2)-c2ccc(OC(F)(F)F)cc2)cc1

InChI Key InChIKey=RGEIPFNQDIMRPC-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50334491   

TargetGlucagon receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334491(3-(4-((3-cyclohexyl-1-(4-(trifluoromethoxy)phenyl)...)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of [125I]glucagon from human GCGR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334491(3-(4-((3-cyclohexyl-1-(4-(trifluoromethoxy)phenyl)...)
Affinity DataIC50:  7.40E+3nMAssay Description:Antagonist activity at human GIPR expressed in CHO cells assessed as inhibition of glucagon-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed