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BDBM50339281 5-(2,6-Dichloro-5-fluoropyridin-3-yl)-3-phenyl-2-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-7(4H)-one::CHEMBL1689654

SMILES: Fc1cc(c(Cl)nc1Cl)-c1cc(=O)n2[nH]c(c(-c3ccccc3)c2n1)C(F)(F)F

InChI Key: InChIKey=ZOLHKPWSDFSDKA-UHFFFAOYSA-N

Data: 2 EC50

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50339281   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Potassium voltage-gated channel subfamily KQT member 2/3


(Human)
BDBM50339281
PNG
(5-(2,6-Dichloro-5-fluoropyridin-3-yl)-3-phenyl-2-(...)
GoogleScholar
UniChem
n/an/an/an/a 60n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily KQT member 1


(Human)
BDBM50339281
PNG
(5-(2,6-Dichloro-5-fluoropyridin-3-yl)-3-phenyl-2-(...)
GoogleScholar
UniChem
n/an/an/an/a 4.93E+4n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair