BDBM50339871 (S)-3-(1-(4-(5-chlorothiophen-2-yl)pyrimidin-2-yl)piperidin-3-yl)-1-ethyl-1H-imidazo[4,5-b]pyridin-2(3H)-one::CHEMBL1761301
SMILES CCn1c2cccnc2n([C@H]2CCCN(C2)c2nccc(n2)-c2ccc(Cl)s2)c1=O
InChI Key InChIKey=LUUJSZJFOWCYDK-AWEZNQCLSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50339871
Affinity DataIC50: 1nMAssay Description:Inhibition of human FAAH assessed as hydrolysis of anandamidoaminomethylcumarinMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Inhibition of FAAH in human T84 cell assessed as conversion of [3H]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 280nMAssay Description:Inhibition of FAAH in rat RBL cell assessed as conversion of [3H]AEA to [3H]ethanolamine by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of rat FAAH assessed as hydrolysis of anandamidoaminomethylcumarinMore data for this Ligand-Target Pair