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BDBM50340729 5,7-Dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidine::CHEMBL1429795::US8552005, 1.1(1)

SMILES: Cc1cc(C)n2ncc(c2n1)S(=O)(=O)c1ccccc1

InChI Key: InChIKey=DERQCQDVQZMDRO-UHFFFAOYSA-N

Data: 3 KI 2 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50340729
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
5-hydroxytryptamine receptor 6 (Human)	BDBM50340729 (CHEMBL1429795 \| US8552005, 1.1(1) \| 5,7-Dimethyl-3...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 6 (Human)	BDBM50340729 (CHEMBL1429795 \| US8552005, 1.1(1) \| 5,7-Dimethyl-3...) Show SMILES Show InChI	GoogleScholar	UniChem		237	n/a	510	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 6 (Human)	BDBM50340729 (CHEMBL1429795 \| US8552005, 1.1(1) \| 5,7-Dimethyl-3...) Show SMILES Show InChI	GoogleScholar	UniChem		237	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 6 (Human)	BDBM50340729 (CHEMBL1429795 \| US8552005, 1.1(1) \| 5,7-Dimethyl-3...) Show SMILES Show InChI	GoogleScholar	UniChem		561	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair