BDBM50374597 CHEMBL271772::US9604926, Compound CM-121::US9724435, Compound CM-121

SMILES O=c1oc2ccccc2n1CCCCN1CCN(CC1)C1CCCCC1

InChI Key InChIKey=WWPDOXILIDUTHY-UHFFFAOYSA-N

Data  9 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50374597   

TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
The University Of Mississippi

US Patent
LigandPNGBDBM50374597(CHEMBL271772 | US9604926, Compound CM-121 | US9724...)
Affinity DataKi:  1.83nMAssay Description:Compounds were evaluated for σ-1 and σ-2 binding in rat brain homogenates. Twelve concentrations of each test ligand (0.001-1,000 nM) were ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Mus musculus (Mouse))
The University Of Mississippi

US Patent
LigandPNGBDBM50374597(CHEMBL271772 | US9604926, Compound CM-121 | US9724...)
Affinity DataKi:  1.83nMAssay Description:Compounds were evaluated for σ-1 and σ-2 binding in rat brain homogenates. Twelve concentrations of each test ligand (0.001-1,000 nM) were ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Mus musculus (Mouse))
The University Of Mississippi

US Patent
LigandPNGBDBM50374597(CHEMBL271772 | US9604926, Compound CM-121 | US9724...)
Affinity DataKi:  1.83nMAssay Description:Compounds were evaluated for σ-1 and σ-2 binding in rat brain homogenates. Twelve concentrations of each test ligand (0.001-1,000 nM) were ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
The University Of Mississippi

US Patent
LigandPNGBDBM50374597(CHEMBL271772 | US9604926, Compound CM-121 | US9724...)
Affinity DataKi:  1.83nMAssay Description:Compounds were evaluated for σ-1 and σ-2 binding in rat brain homogenates. Twelve concentrations of each test ligand (0.001-1,000 nM) were ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by PDSP Ki Database
LigandPNGBDBM50374597(CHEMBL271772 | US9604926, Compound CM-121 | US9724...)
Affinity DataKi:  11.3nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
The University Of Mississippi

US Patent
LigandPNGBDBM50374597(CHEMBL271772 | US9604926, Compound CM-121 | US9724...)
Affinity DataKi:  11.3nMAssay Description:Compounds were evaluated for σ-1 and σ-2 binding in rat brain homogenates. Twelve concentrations of each test ligand (0.001-1,000 nM) were ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by PDSP Ki Database
LigandPNGBDBM50374597(CHEMBL271772 | US9604926, Compound CM-121 | US9724...)
Affinity DataKi:  11.3nMAssay Description:Compounds were evaluated for σ-1 and σ-2 binding in rat brain homogenates. Twelve concentrations of each test ligand (0.001-1,000 nM) were ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
The University Of Mississippi

US Patent
LigandPNGBDBM50374597(CHEMBL271772 | US9604926, Compound CM-121 | US9724...)
Affinity DataKi:  11.3nMAssay Description:Compounds were evaluated for σ-1 and σ-2 binding in rat brain homogenates. Twelve concentrations of each test ligand (0.001-1,000 nM) were ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by PDSP Ki Database
LigandPNGBDBM50374597(CHEMBL271772 | US9604926, Compound CM-121 | US9724...)
Affinity DataKi:  11.3nMAssay Description:Compounds were evaluated for σ-1 and σ-2 binding in rat brain homogenates. Twelve concentrations of each test ligand (0.001-1,000 nM) were ...More data for this Ligand-Target Pair
In DepthDetails US Patent