BDBM50395136 CHEMBL2163965

SMILES O=C(NC1CCCC1)c1cn2C(COc3cccc(c23)c1=O)c1ccccc1

InChI Key InChIKey=FKTORJCFBBTXPW-UHFFFAOYSA-N

Data  4 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50395136   

TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£ di Ferrara

Curated by ChEMBL
LigandPNGBDBM50395136(CHEMBL2163965)
Affinity DataKi:  98nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in CHO cell membranes incubated for 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Universit£ di Ferrara

Curated by ChEMBL
LigandPNGBDBM50395136(CHEMBL2163965)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in Sprague-Dawley rat spleen by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£ di Ferrara

Curated by ChEMBL
LigandPNGBDBM50395136(CHEMBL2163965)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in CHO cell membranes incubated for 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universit£ di Ferrara

Curated by ChEMBL
LigandPNGBDBM50395136(CHEMBL2163965)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat brain by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£ di Ferrara

Curated by ChEMBL
LigandPNGBDBM50395136(CHEMBL2163965)
Affinity DataIC50:  472nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cell membranes assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed