BDBM50399656 CHEMBL2069623::US11633415, Compound PF4800567
SMILES Nc1ncnc2n(nc(COc3cccc(Cl)c3)c12)C1CCOCC1
InChI Key InChIKey=AUMDBEHGJRZSOO-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 50399656
Affinity DataIC50: 711nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of CK1epsilonMore data for this Ligand-Target Pair
Affinity DataIC50: 711nMAssay Description:Inhibition of Casein kinase 1 deltaMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of Casein kinase 1 epsilonMore data for this Ligand-Target Pair
Affinity DataIC50: 857nMAssay Description:In order to identify inhibitors of CSNK1A1, the CSNK1A1 knockdown signatures in CMap were compared to all CMap compound signatures, and resultant com...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of human full length CK1delta1 (2 to 415 residues) using PLSRTLpSVASLPGL as substrate after 2 hrs by kinase-glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 711nMAssay Description:Inhibition of human CK1delta in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of human CK1epsilon in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of human full length polyhistidine-tagged CK1epsilon expressed in Escherichia coli BL21-Codon-Plus (DE3)-RIL using PLSRTLpSVASLPGL as subs...More data for this Ligand-Target Pair