BDBM50399838 CHEMBL2180285

SMILES CCCC1=C(C(C2C(=O)CC(C)(C)CC2=N1)c1ccc(cc1)-c1ccccc1)C(=O)OCC

InChI Key InChIKey=MPVREJOAMJGRQF-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50399838   

TargetTGF-beta receptor type-2(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50399838(CHEMBL2180285)
Affinity DataIC50:  830nMAssay Description:Inhibition of TGBR2 signaling in human HEK293T cells assessed as inhibition of SMAD activation after 2 to 22 hrs by dual Luciferase AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed