BDBM50418189 CHEMBL1761696

SMILES C[C@H](NCc1c(noc1-c1ccc(cc1)C(F)(F)F)C(=O)N[C@@H]1CCC[C@H](O)C1)C(F)(F)F

InChI Key InChIKey=NNEPHZMMSYMBQT-GLQYFDAESA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50418189   

TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Msd

Curated by ChEMBL

LigandBDBM50418189(CHEMBL1761696)Copy SMILESCopy InChI

Affinity DataIC50:  0.158nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO-K1 cells assessed as inhibition of capsaicin-induced intracellular Ca2+ influx by FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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