BDBM50430605 CHEMBL2338715::Rel-Ethylketazocine
SMILES CC[C@]12CCN(CC3CC3)[C@H]([C@H]1C)C(=O)c1ccc(O)cc21
InChI Key InChIKey=SEJUQQOPVAUETF-LLSQANQASA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50430605
Affinity DataKi: 0.390nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20nMAssay Description:Agonist activity at human KOR expressed in CHO cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 4.40nMAssay Description:Agonist activity at rat recombinant MOR expressed in rat C6 cells assessed as stimulation of [35S]GTPgammaS binding after 1 hrMore data for this Ligand-Target Pair