BDBM50430802 CHEMBL2334775

SMILES Cc1cc(O)cc(C)c1C[C@H](N)C(=O)N1CC[C@@H](C1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](C(=C)C(N)=O)c1ccco1

InChI Key InChIKey=RIAOSVMITNWHAH-HFASDWQVSA-N

Data  3 KI  2 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 50430802   

TargetMu-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50430802(CHEMBL2334775)
Affinity DataKi:  0.0128nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50430802(CHEMBL2334775)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]DPDPE from Myc-tagged delta-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50430802(CHEMBL2334775)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]U69,593 from kappa-type opioid receptor (unknown origin) expressed in HEK293 cells after 60 mins by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50430802(CHEMBL2334775)
Affinity DataIC50:  0.834nMAssay Description:Agonist activity at mu-type opioid receptor in guinea pig ileum assessed as inhibition of electrically evoked muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50430802(CHEMBL2334775)
Affinity DataEC50:  47nMAssay Description:Agonist activity at Myc-tagged delta-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50430802(CHEMBL2334775)
Affinity DataEC50:  0.000109nMAssay Description:Agonist activity at FLAG-tagged mu-type opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50430802(CHEMBL2334775)
Affinity DataIC50:  0.962nMAssay Description:Agonist activity at mu-type opioid receptor in Kunming mouse vas deferens assessed as inhibition of electrically evoked muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed