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BDBM50434338 CHEMBL2386762::US9446044, 56

SMILES: COC(=N)c1nc2ccc3ncnc(Nc4ccc(Cl)cc4)c3c2s1

InChI Key: InChIKey=BGXZIBSLBRKDTP-UHFFFAOYSA-N

Data: 4 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50434338
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Dual specificity tyrosine-phosphorylation-regulated kinase 1A (Human)	BDBM50434338 (CHEMBL2386762 \| US9446044, 56) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.13	n/a	n/a	n/a	n/a	7.5	25
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Dual specificity tyrosine-phosphorylation-regulated kinase 1B (Human)	BDBM50434338 (CHEMBL2386762 \| US9446044, 56) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	4.74	n/a	n/a	n/a	n/a	7.5	25
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Dual specificity tyrosine-phosphorylation-regulated kinase 1B (Human)	BDBM50434338 (CHEMBL2386762 \| US9446044, 56) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	4.70	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Dual specificity tyrosine-phosphorylation-regulated kinase 1A (Human)	BDBM50434338 (CHEMBL2386762 \| US9446044, 56) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.10	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair