BDBM50440059 CHEMBL2426082

SMILES OC(=O)CCC(=O)N1N=C(C[C@@H]1c1ccc(Cl)cc1)c1c(-c2ccc(Cl)cc2)c2ccccc2[nH]c1=O

InChI Key InChIKey=PXQFOMCFQUXMBP-HSZRJFAPSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50440059   

TargetGlutamate receptor ionotropic, NMDA 2D(Rattus norvegicus (Rat))
Emory University

Curated by ChEMBL
LigandPNGBDBM50440059(CHEMBL2426082)
Affinity DataIC50:  1.90E+3nMAssay Description:Negative allosteric modulation of recombinant rat GluN2D receptor expressed in Xenopus laevis oocytes by two-electrode voltage clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2A(Rattus norvegicus (Rat))
Emory University

Curated by ChEMBL
LigandPNGBDBM50440059(CHEMBL2426082)
Affinity DataIC50:  4.50E+4nMAssay Description:Negative allosteric modulation of recombinant rat GluN2A receptor expressed in Xenopus laevis oocytes by two-electrode voltage clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Emory University

Curated by ChEMBL
LigandPNGBDBM50440059(CHEMBL2426082)
Affinity DataIC50:  5.20E+4nMAssay Description:Negative allosteric modulation of recombinant rat GluN2B receptor expressed in Xenopus laevis oocytes by two-electrode voltage clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
Emory University

Curated by ChEMBL
LigandPNGBDBM50440059(CHEMBL2426082)
Affinity DataIC50:  2.10E+3nMAssay Description:Negative allosteric modulation of recombinant rat GluN2C receptor expressed in Xenopus laevis oocytes by two-electrode voltage clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed