BDBM50443584 CHEMBL3091980
SMILES CN(C1C[C@@H]2CCCC[C@@H]2[C@H]1\C=C\c1ccc(cn1)-c1cccc(F)c1)S(C)(=O)=O
InChI Key InChIKey=BRSCNTKXIWSLQX-DKBLXCOBSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50443584
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Korea Research Institute Of Technology
Curated by ChEMBL
Korea Research Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Antagonist activity at PAR1 in human platelet rich plasma assessed as inhibition of haTRAP-induced platelet aggregation preincubated for 1 hr followe...More data for this Ligand-Target Pair
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Korea Research Institute Of Technology
Curated by ChEMBL
Korea Research Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]haTRAP from PAR1 in human platelet membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Korea Research Institute Of Technology
Curated by ChEMBL
Korea Research Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at PAR1 in washed human platelets assessed as inhibition of haTRAP-induced platelet aggregation preincubated for 1 hr followed by...More data for this Ligand-Target Pair