BDBM50455155 CHEMBL4217737

SMILES Fc1cc(c(F)cc1OC[C@H]1OCCN[C@@H]1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1

InChI Key InChIKey=IEAKVRVAJJXUBH-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50455155   

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50455155(CHEMBL4217737)
Affinity DataIC50: 2.90E+4nMAssay Description:Antagonist activity at recombinant human Nav1.7 expressed in HEK293 cells assessed as reduction in channel current at -60 mV holding potential after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed