BDBM50494191 CHEMBL3086094

SMILES O=C(c1nc2ccccc2[nH]1)c1ccc(Oc2nccnc2N2CCCOCC2)cc1

InChI Key InChIKey=FSOBJGLZSZGYOL-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50494191   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Amgen

Curated by ChEMBL

LigandBDBM50494191(CHEMBL3086094)Copy SMILESCopy InChI

Affinity DataIC50: 5.10nMAssay Description:Inhibition of human recombinant PDE10A using cAMP as substrate preincubated for 30 mins prior to substrate addition measured after 1 hr by IMAP TR-FR...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
9/1/2020
Entry Details Article
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