BDBM50513125 CHEMBL4440510

SMILES COC(=O)c1ccc2c(C(CC(F)(F)F)c3cccs3)c([nH]c2c1)-c1ccccc1

InChI Key InChIKey=MMQZODPLDCMCIS-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50513125   

TargetCannabinoid receptor 1(Human)
University of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50513125(CHEMBL4440510)
Affinity DataEC50:  160nMAssay Description:Positive allosteric modulation of human CB1 receptor expressed in CHOK1 cells assessed as increase in CP55940-induced beta-arrestin recruitment prein...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50513125(CHEMBL4440510)
Affinity DataEC50:  160nMAssay Description:Positive allosteric modulation of human CB1 receptor expressed in CHOK1 cells assessed as increase in CP55940-induced beta-arrestin recruitment prein...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50513125(CHEMBL4440510)
Affinity DataEC50:  682nMAssay Description:Agonist activity at human CB1 receptor expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 30 mins by PathHunt...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50513125(CHEMBL4440510)
Affinity DataEC50:  682nMAssay Description:Agonist activity at human CB1 receptor expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 30 mins by PathHunt...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed