BDBM50527380 CHEMBL4517118

SMILES CCOc1cc(c(c(c1)C(=O)NNS(=O)(=O)c2ccc3ccccc3c2)F)C

InChI Key InChIKey=ZHPGBCFNKHBCKG-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50527380   

TargetHistone acetyltransferase KAT6A [507-778](Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50527380(CHEMBL4517118)
Affinity DataIC50: 82nMAssay Description:Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed