BDBM50529873 CHEMBL4552616
SMILES Cc1ncccc1Oc1sc(C(N)=O)c2CCc3cnn(C)c3-c12
InChI Key InChIKey=IUIDISNVIBKQQL-UHFFFAOYSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50529873
Affinity DataIC50: 1.60nMAssay Description:Displacement of Kinase tracer 236 from recombinant full-length human N-terminal GST-fused CDK8 (1 to 464 residues)/cyclin C (1 to 283 residues) expre...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Displacement of Kinase tracer 236 from GST-fused CDK19/cyclin C (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Displacement of Kinase tracer 236 from recombinant full-length human N-terminal GST-fused CDK8 (1 to 464 residues)/cyclin C (1 to 283 residues) expre...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Displacement of Kinase tracer 236 from GST-fused CDK19/cyclin C (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair