Found 107 hits for monomerid = 517 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Dimer of Gag-Pol polyprotein [501-599]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 0.360 | n/a | n/a | n/a | n/a | 5.5 | 30 |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Dimer of Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 0.360 | n/a | n/a | n/a | n/a | 5.5 | 30 |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Dimer of Gag-Pol polyprotein [489-587,Q496K]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 0.590 | n/a | n/a | n/a | n/a | 5.5 | 30 |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Dimer of Gag-Pol polyprotein [489-587,Q496K]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a | 5.5 | 30 |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Dimer of Gag-Pol polyprotein [489-587,Q496K,L499I,M525I,N526D,M535I,R546K,L552P,A560V,G562S,I573V,L579M,I582L]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 61 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Dimer of Gag-Pol polyprotein [489-587,Q496K]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a | 5.5 | 30 |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Dimer of Gag-Pol polyprotein [489-587,Q496K,L499I,M535I,I543V,Q547E,L552P,I553V,V566I,V571F,I573V,L579M,I582L]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 61.2 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Dimer of Gag-Pol polyprotein [489-587,Q496K,L499I,M525I,N526D,M535I,R546K,L552P,A560V,G562S,I573V,L579M,I582L]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 43.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Dimer of Gag-Pol polyprotein [489-587,Q496K,L499I,N526S,R530K,M535I,I543V,I551V,L552P,A560V,V566I,V571A,L579M,I582L]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 20.1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Dimer of Gag-Pol polyprotein [489-587,Q496K]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a | 5.5 | 30 |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Dimer of Gag-Pol polyprotein [489-587,Q496K,L499I,M535I,I543V,Q547E,L552P,I553V,V566I,V571F,I573V,L579M,I582L]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 61.2 | n/a | n/a | n/a | n/a | 5.5 | 30 |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Dimer of Gag-Pol polyprotein [489-587,Q496K,L499I,M525I,N526D,M535I,R546K,L552P,A560V,G562S,I573V,L579M,I582L]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 43.6 | n/a | n/a | n/a | n/a | 5.5 | 30 |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Dimer of Gag-Pol polyprotein [489-587,Q496K,L499I,N526S,R530K,M535I,I543V,I551V,L552P,A560V,V566I,V571A,L579M,I582L]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 20.1 | n/a | n/a | n/a | n/a | 5.5 | 30 |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag polyprotein
(HIV-1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 20 | n/a | n/a | n/a | n/a | 6.5 | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 0.560 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 0.590 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 89 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.60 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 0.590 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 0.590 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Cytochrome P450 3A4
(Human) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Cytochrome P450 2D6
(Human) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 61 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 0.410 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 370 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 0.360 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 0.590 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 0.410 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 52 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 56 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | n/a | n/a | n/a | 0.00158 | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | n/a | 1.07 | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
ATP-dependent translocase ABCB1
(Human) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
ATP-dependent translocase ABCB1
(Human) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 4.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Multidrug and toxin extrusion protein 2
(Human) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Multidrug and toxin extrusion protein 1
(Human) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 7.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Multidrug and toxin extrusion protein 2
(Human) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 7.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Solute carrier family 22 member 3
(Human) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Solute carrier family 22 member 1
(Human) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 2.08E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Solute carrier family 22 member 2
(Human) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.42E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Multidrug and toxin extrusion protein 1
(Human) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Multidrug and toxin extrusion protein 1
(Human) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Dimer of Gag-Pol polyprotein [489-587,V571I]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | 0.0520 | -14.3 | n/a | n/a | n/a | n/a | n/a | 5.5 | 30 |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Dimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | 0.0700 | -13.8 | n/a | n/a | n/a | n/a | n/a | 6.4 | 25 |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Dimer of Gag-Pol polyprotein [489-587,L565M]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | 0.114 | -13.8 | n/a | n/a | n/a | n/a | n/a | 5.5 | 30 |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | 0.240 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Gag-Pol polyprotein [489-587]
(Human immunodeficiency virus type 1) | BDBM517
 (Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...) | GoogleScholar
| UniChem
| | 0.280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |