BDBM564474 Roche-Dataset for PDE10A, Compound 788

SMILES c1cc2c(cc1NC(=O)c3c(ccc(n3)C4CC4)Nc5cncnc5)C(=O)NC2

InChI Key InChIKey=IDHJZGWRFDFBHP-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 564474   

LigandPNGBDBM564474(Roche-Dataset for PDE10A, Compound 788)
Affinity DataIC50: 20nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed