Found 13 hits for monomerid = 7534 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Cyclin-dependent kinase 1/G2/mitotic-specific cyclin-B
(Spiny starfish) | BDBM7534
 (1H-pyrazolo[3,4-b]quinoxalin-3-amine | pyrazolo[3,...) | GoogleScholar
| UniChem
| | n/a | n/a | 600 | n/a | n/a | n/a | n/a | 7.2 | 30 |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Cyclin-dependent kinase/G2/mitotic-specific cyclin- 1
(Human) | BDBM7534
 (1H-pyrazolo[3,4-b]quinoxalin-3-amine | pyrazolo[3,...) | GoogleScholar
| UniChem
| | n/a | n/a | 9.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Cyclin-A2/Cyclin-dependent kinase 2
(Human) | BDBM7534
 (1H-pyrazolo[3,4-b]quinoxalin-3-amine | pyrazolo[3,...) | GoogleScholar
| UniChem
| | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Cyclin-dependent kinase 4/G1/S-specific cyclin-D1
(Human) | BDBM7534
 (1H-pyrazolo[3,4-b]quinoxalin-3-amine | pyrazolo[3,...) | GoogleScholar
| UniChem
| | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Cyclin-dependent kinase 5 activator 1
(Human) | BDBM7534
 (1H-pyrazolo[3,4-b]quinoxalin-3-amine | pyrazolo[3,...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.37E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
CDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7
(Human) | BDBM7534
 (1H-pyrazolo[3,4-b]quinoxalin-3-amine | pyrazolo[3,...) | GoogleScholar
| UniChem
| | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Cyclin-T1/Cyclin-dependent kinase 9
(Human) | BDBM7534
 (1H-pyrazolo[3,4-b]quinoxalin-3-amine | pyrazolo[3,...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.41E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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More data for this Ligand-Target Pair | |
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1
(Human) | BDBM7534
 (1H-pyrazolo[3,4-b]quinoxalin-3-amine | pyrazolo[3,...) | GoogleScholar
| UniChem
| | n/a | n/a | 5.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Cyclin-dependent kinase 5 activator 1
(Human) | BDBM7534
 (1H-pyrazolo[3,4-b]quinoxalin-3-amine | pyrazolo[3,...) | GoogleScholar
| UniChem
| | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Human) | BDBM7534
 (1H-pyrazolo[3,4-b]quinoxalin-3-amine | pyrazolo[3,...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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More data for this Ligand-Target Pair | |
Interferon-induced, double-stranded RNA-activated protein kinase
(Human) | BDBM7534
 (1H-pyrazolo[3,4-b]quinoxalin-3-amine | pyrazolo[3,...) | GoogleScholar
| UniChem
| | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Human) | BDBM7534
 (1H-pyrazolo[3,4-b]quinoxalin-3-amine | pyrazolo[3,...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Cyclin-dependent kinase 1/G2/mitotic-specific cyclin-B1/G2/mitotic-specific cyclin-B2/G2/mitotic-specific cyclin-B3
(Human) | BDBM7534
 (1H-pyrazolo[3,4-b]quinoxalin-3-amine | pyrazolo[3,...) | GoogleScholar
| UniChem
| | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |