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BDBM81467 CAS_569-65-3::CHEMBL1085765::Meclizine::NSC_4034::US9182402, 13

SMILES: Cc1cccc(CN2CCN(CC2)C(c2ccccc2)c2ccc(Cl)cc2)c1

InChI Key: InChIKey=OCJYIGYOJCODJL-UHFFFAOYSA-N

Data: 1 KI 5 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 81467
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Serine protease hepsin (Human)	BDBM81467 (CHEMBL1085765 \| NSC_4034 \| CAS_569-65-3 \| Meclizin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.02E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Trypsin (Pig)	BDBM81467 (CHEMBL1085765 \| NSC_4034 \| CAS_569-65-3 \| Meclizin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Prothrombin (Bovine)	BDBM81467 (CHEMBL1085765 \| NSC_4034 \| CAS_569-65-3 \| Meclizin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cruzipain (Trypanosoma cruzi)	BDBM81467 (CHEMBL1085765 \| NSC_4034 \| CAS_569-65-3 \| Meclizin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.29E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cruzipain (Trypanosoma cruzi)	BDBM81467 (CHEMBL1085765 \| NSC_4034 \| CAS_569-65-3 \| Meclizin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>2.50E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Histamine H1 receptor (Rat)	BDBM81467 (CHEMBL1085765 \| NSC_4034 \| CAS_569-65-3 \| Meclizin...) Show SMILES Show InChI	GoogleScholar	UniChem		250	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair