BDBM82376 CAS_80880-90-6::NSC_5387::TELENZEPINE

SMILES: CN1CCN(CC(=O)N2c3c(C)scc3C(=O)Nc3ccccc23)CC1

InChI Key: InChIKey=VSWPGAIWKHPTKX-UHFFFAOYSA-N

Data: 12 KI  1 IC50

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 13 hits for monomerid = 82376   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Bile salt export pump (Human)	BDBM82376 (NSC_5387 | CAS_80880-90-6 | TELENZEPINE) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.15E+5	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1 (Rat)	BDBM82376 (NSC_5387 | CAS_80880-90-6 | TELENZEPINE) Show SMILES Show InChI	GoogleScholar	UniChem		1.29	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1 (Rat)	BDBM82376 (NSC_5387 | CAS_80880-90-6 | TELENZEPINE) Show SMILES Show InChI	GoogleScholar	UniChem		1.80	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M4 (Chicken)	BDBM82376 (NSC_5387 | CAS_80880-90-6 | TELENZEPINE) Show SMILES Show InChI	GoogleScholar	UniChem		2.45	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor (Rabbit)	BDBM82376 (NSC_5387 | CAS_80880-90-6 | TELENZEPINE) Show SMILES Show InChI	GoogleScholar	UniChem		2.63	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M4 (Bovine)	BDBM82376 (NSC_5387 | CAS_80880-90-6 | TELENZEPINE) Show SMILES Show InChI	GoogleScholar	UniChem		5.88	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M3 (Rat)	BDBM82376 (NSC_5387 | CAS_80880-90-6 | TELENZEPINE) Show SMILES Show InChI	GoogleScholar	UniChem		6.90	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M3 (Rat)	BDBM82376 (NSC_5387 | CAS_80880-90-6 | TELENZEPINE) Show SMILES Show InChI	GoogleScholar	UniChem		7.59	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor (Pig)	BDBM82376 (NSC_5387 | CAS_80880-90-6 | TELENZEPINE) Show SMILES Show InChI	GoogleScholar	UniChem		12.6	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M2 (Rat)	BDBM82376 (NSC_5387 | CAS_80880-90-6 | TELENZEPINE) Show SMILES Show InChI	GoogleScholar	UniChem		17.0	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M4 (Rat)	BDBM82376 (NSC_5387 | CAS_80880-90-6 | TELENZEPINE) Show SMILES Show InChI	GoogleScholar	UniChem		17	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M2 (Rat)	BDBM82376 (NSC_5387 | CAS_80880-90-6 | TELENZEPINE) Show SMILES Show InChI	GoogleScholar	UniChem		50	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M4 (Rat)	BDBM82376 (NSC_5387 | CAS_80880-90-6 | TELENZEPINE) Show SMILES Show InChI	GoogleScholar	UniChem		67.6	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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