BDBM85515 Ampyrone::CAS_83-07-8::EN300-17058::NSC_2151::US11643395, Compound 9
SMILES Cc1c(N)c(=O)n(-c2ccccc2)n1C
InChI Key InChIKey=RLFWWDJHLFCNIJ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 85515
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of COX-1 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 6.97E+4nMAssay Description:In-vitro butyryl cholinesterase inhibitory activity was performed in 96-well microplates, 0.5 mM test compound in methanol, was incubated with 20 ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of COX-2 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 3.41E+3nMAssay Description:IC50 values were determined for the whole plate in case of Chan-Lam coupling, using 5 point 3-fold dilutions (starting from 10 μM).More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of purified ovine COX1 pre-treated for 1 hr before 10-acetyl-3,7-dihydroxyphenoxazin substrate addition in absence of porcine liver estera...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of human recombinant COX2 pre-treated for 1 hr before 10-acetyl-3,7-dihydroxyphenoxazin substrate addition in absence of porcine liver est...More data for this Ligand-Target Pair