BDBM85830 VUF5202

SMILES Clc1ccc(CNCCCCCc2cnc[nH]2)cc1

InChI Key InChIKey=BJZMQYYHQDWJRH-UHFFFAOYSA-N

Data  1 KI  1 IC50  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 85830   

TargetHistamine H3 receptor(Homo sapiens (Human))
Vrije Universiteit

Curated by PDSP Ki Database
LigandPNGBDBM85830(VUF5202)
Affinity DataKi:  2.34nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H3 receptor(GUINEA PIG)
De Novo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM85830(VUF5202)
Affinity DataKd:  1.26nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptors in homogenates of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vrije Universiteit

Curated by PDSP Ki Database
LigandPNGBDBM85830(VUF5202)
Affinity DataIC50:  1.30nMAssay Description:Activity against human H3 receptor as measured by CRE-mediated beta galactosidase reporter gene assay in forskolin-stimulated SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed